The order of decreasing reactivity towards an electrophilic reagent, for the following would be: (i) benzene…

The order of decreasing reactivity towards an electrophilic reagent, for the following would be: (i) benzene (ii) toluene (iii) chlorobenzene (iv) phenol
  1. (ii) $ > $ (iv) $ > $ (i) $ > $ (iii)
  2. (iv) $ > $ (iii) $ > $ (ii) $ > $ (i)
  3. (iv) $ > $ (ii) $ > $ (i) $ > $ (iii)
  4. (i) $ > $ (ii) $ > $ (iii) $ > $ (iv)

Solution

Electrophiles have high affinity for electrons. They attack at the site where electron-density is highest. Electron withdrawing substances increases the electron density. The electron withdrawing tendency decreases in the order : $-\mathrm{OH} > -\mathrm{CH}_3 > -\mathrm{H} > -\mathrm{Cl}$ Therefore, the correct order of reactivity towards electrophile is $\mathrm{C}_6 \mathrm{H}_5 \mathrm{OH} > \mathrm{C}_6 \mathrm{H}_5 \mathrm{CH}_3 > \mathrm{C}_6 \mathrm{H}_6 > \mathrm{C}_6 \mathrm{H}_5 \mathrm{Cl}$ Related Theory Electrophilic substitution reaction in haloarenes occur slowly because halogen has a negative inductive effect, it decreases the electron density on the benzene ring due to resonance.

Asked in: NEET 2007

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